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authIdHal_s : caroline-barette
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Les criblages phénotypiques ou comment faire d’une pierre deux coups

Renaud Prudent , Emmanuelle Soleilhac , Caroline Barette , Marie-Odile Fauvarque , Laurence Lafanechère
Médecine/Sciences, 2013, 29 (10), pp.897-905. ⟨10.1051/medsci/20132910018⟩
Journal articles hal-03095110v1

Single assay-wide variance experimental (SAVE) design for high-throughput screening

Carl Murie , Caroline Barette , Laurence Lafanechère , Robert Nadon
Bioinformatics, 2013, 29 (23), pp.3067-3072. ⟨10.1093/bioinformatics/btt538⟩
Journal articles hal-02347938v1

High-Content Screening Identifies New Inhibitors of Connexin 43 Gap Junctions

Christèle Picoli , Emmanuelle Soleilhac , Agnès Journet , Caroline Barette , Marjorie Comte , et al.
ASSAY and Drug Development Technologies, 2019, 17 (5), pp.240-248. ⟨10.1089/adt.2019.927⟩
Journal articles hal-02284993v1
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Compounds with antiparasitic activity and applications thereof

Djeneb Camara , Cordelia Bisanz , Caroline Barette , Marie-France Cesbron-Delauw , Fabrice Rébeillé
Patent n° : 11290215.0 - 1211. 2011, 18 p
Patents hal-00790622v1
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Inhibition of p-Aminobenzoate and Folate Syntheses in Plants and Apicomplexan Parasites by Natural Product Rubreserine.

Djeneb Camara , Cordelia Bisanz , Caroline Barette , Jeroen van Daele , Esmare Human , et al.
Journal of Biological Chemistry, 2012, 287 (26), pp.22367-76. ⟨10.1074/jbc.M112.365833⟩
Journal articles hal-00702251v1

Control-Plate Regression (CPR) Normalization for High-Throughput Screens with Many Active Features

C. Murie , C. Barette , L. Lafanechère , R. Nadon
Journal of Biomolecular Screening, 2014, 19 (5), pp.661-671. ⟨10.1177/1087057113516003⟩
Journal articles hal-02177825v1

Synthesis and biological evaluation of thiophene and benzo[b]thiophene analogs of combretastatin A-4 and isocombretastatin A-4: A comparison between the linkage positions of the 3,4,5-trimethoxystyrene unit

Cong Viet Do , Abdelfattah Faouzi , Caroline Barette , Amaury Farce , Marie-Odile Fauvarque , et al.
Bioorganic and Medicinal Chemistry Letters, 2016, 26 (1), pp.174-180. ⟨10.1016/j.bmcl.2015.11.010⟩
Journal articles hal-02176934v1
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Investigation of chemical composition and biological activities of $Ajuga\ pyramidalis$—isolation of iridoids and phenylethanoid glycosides

Anthonin Gori , Benjamin Boucherle , Aurélien Rey , Maxime Rome , Caroline Barette , et al.
Metabolites, 2023, 13, pp.128. ⟨10.3390/metabo13010128⟩
Journal articles hal-04014499v1

Identification of polyoxometalates as nanomolar noncompetitive inhibitors of protein kinase CK2.

Renaud Prudent , Virginie Moucadel , Béatrice Laudet , Caroline Barette , Laurence Lafanechère , et al.
Chemistry & Biology / Chemistry and Biology; CHEMISTRY & BIOLOGY, 2008, 15 (7), pp.683-92. ⟨10.1016/j.chembiol.2008.05.018⟩
Journal articles hal-00345731v1

Functional characterization of cell-free expressed K v 1.3 channel using a voltage-sensitive fluorescent dye

Sandra Cortès , Caroline Barette , Rémy Beroud , Michel de Waard , Béatrice Schaack
Protein Expression and Purification, 2018, 145, pp.94 - 99. ⟨10.1016/j.pep.2018.01.006⟩
Journal articles hal-01726204v1

Screening for Biologically Annotated Drugs That Trigger Triacylglycerol Accumulation in the Diatom Phaeodactylum

Melissa Conte , Josselin Lupette , Khawla Seddiki , Coline Meï , Lina-Juana Dolch , et al.
Plant Physiology, 2018, 177 (2), pp.532 - 552. ⟨10.1104/pp.17.01804⟩
Journal articles hal-01851869v1
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Acacetin and Chrysin, Two Polyphenolic Compounds, Alleviate Telomeric Position Effect in Human Cells

Amina Boussouar , Caroline Barette , Robert Nadon , Adelaïde Saint-Léger , Natacha Broucqsault , et al.
Molecular Therapy - Nucleic Acids, 2013, 2, pp.e116. ⟨10.1038/mtna.2013.42⟩
Journal articles hal-01617538v1

Improving Detection of Rare Biological Events in High-Throughput Screens

Carl Murie , Caroline Barette , Jennifer Button , Laurence Lafanechere , Robert Nadon
Journal of Biomolecular Screening, 2015, 20 (2), pp.230-241. ⟨10.1177/1087057114548853⟩
Journal articles hal-02176981v1

Criblages phénotypiques et génétique chimique directe. Une approche innovante pour la découverte de molécules bio-actives et / ou de candidats-médicaments

E. Sans-Soleilhac , C. Barette , S. Wieczorek , Sylvaine Roy , Eric Maréchal , et al.
Spectra Analyse, 2003, 32 (233), pp.33-37
Journal articles hal-02679732v1

Azaindole derivatives are inhibitors of microtubule dynamics, with anti-cancer and anti-angiogenic activities

R. Prudent , E. Vassal-Stermann , Chi-Hung Nguyen , M. Mollaret , J. Viallet , et al.
British Journal of Pharmacology, 2013, 168 (3), pp.673-685. ⟨10.1111/j.1476-5381.2012.02230.x⟩
Journal articles hal-00777455v1

Novel synthetic pharmacophores inducing a stabilization of cellular microtubules

Anne Martinez , Emmanuelle Soleilhac , Caroline Barette , Renaud Prudent , Gustavo Gozzi , et al.
Current Cancer Drug Targets, 2015, 15 (1), pp.2-13. ⟨10.2174/1568009615666141215154149⟩
Journal articles hal-02176978v1

Human cyclin C protein is stabilized by its associated kinase cdk8, independently of its catalytic activity

C. Barette , I. Jariel-Encontre , Marc Piechaczyk , J. Piette
Oncogene, 2001, 20 (5), pp.551--62. ⟨10.1038/sj.onc.1204129⟩
Journal articles hal-02197302v1

Quantitative Automated Assays in Living Cells to Screen for Inhibitors of Hemichannel Function

Emmanuelle Soleilhac , Marjorie Comte , Anaelle da Costa , Caroline Barette , Christèle Picoli , et al.
Slas Discovery, 2020, pp.247255522095438. ⟨10.1177/2472555220954388⟩
Journal articles hal-03093762v1
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A New Quantitative Cell-Based Assay Reveals Unexpected Microtubule Stabilizing Activity of Certain Kinase Inhibitors, Clinically Approved or in the Process of Approval

Sacnicte Ramirez-Rios , Sophie Michallet , Leticia Peris , Caroline Barette , Clotilde Rabat , et al.
Frontiers in Pharmacology, 2020, 11, ⟨10.3389/fphar.2020.00543⟩
Journal articles hal-03034431v1
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Chimeric Protein–Protein Interface Inhibitors Allow Efficient Inhibition of Type III Secretion Machinery and Pseudomonas aeruginosa Virulence

Tuan-Dung Ngo , Sophie Plé , Aline Thomas , Caroline Barette , Antoine Fortuné , et al.
ACS Infectious Diseases, 2019, 5 (11), pp.1843-1854. ⟨10.1021/acsinfecdis.9b00154⟩
Journal articles hal-02318760v1

Isoconazole and Clemizole Hydrochloride Partially Reverse the Xeroderma Pigmentosum C Phenotype

Farah Kobaisi , Eric Sulpice , Caroline Barette , Nour Fayyad , Marie-Odile Fauvarque , et al.
International Journal of Molecular Sciences, 2021, 22 (15), pp.8156. ⟨10.3390/ijms22158156⟩
Journal articles hal-03656560v1
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Identification of chemicals breaking the USP8 interaction with its endocytic substrate CHMP1B

Agnès Journet , Caroline Barette , Laurence Aubry , Emmanuelle Soleilhac , Marie-Odile Fauvarque
Slas Discovery, 2022, 27 (7), pp.395-404. ⟨10.1016/j.slasd.2022.08.003⟩
Journal articles hal-03853845v1
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Cytidine deaminase deficiency in tumor cells is associated with sensitivity to a naphthol derivative and a decrease in oncometabolite levels

Hamza Mameri , Géraldine Buhagiar-Labarchède , Gaëlle Fontaine , Céline Corcelle , Caroline Barette , et al.
Cellular and Molecular Life Sciences, 2022, 79 (8), pp.465. ⟨10.1007/s00018-022-04487-9⟩
Journal articles hal-03766208v1

A new chemical inhibitor of angiogenesis and tumorigenesis that targets the VEGF signaling pathway upstream of Ras

Agnès Desroches-Castan , Delphine Quélard , Martine Demeunynck , Jean-François Constant , Chongling Dong , et al.
Oncotarget, 2015, 6 (7), ⟨10.18632/oncotarget.2979⟩
Journal articles hal-02176957v1
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Cooperative Blockade of CK2 and ATM Kinases Drives Apoptosis in VHL-Deficient Renal Carcinoma Cells through ROS Overproduction

Sofia Giacosa , Catherine Pillet , Irinka Séraudie , Laurent Guyon , Yann Wallez , et al.
Cancers, 2021, 13 (3), pp.576. ⟨10.3390/cancers13030576⟩
Journal articles hal-03134709v1

Miniaturization and Validation of a Sensitive Multiparametric Cell-Based Assay for the Concomitant Detection of Microtubule-Destabilizing and Microtubule-Stabilizing Agents

Emilie Vassal , Caroline Barette , Xavier Fonrose , Raphaël Dupont , Emmanuelle Sans-Soleilhac , et al.
Journal of Biomolecular Screening, 2006, 11 (4), pp.377-389. ⟨10.1177/1087057106286210⟩
Journal articles hal-02348186v1
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Structure-based design of small peptide inhibitors of protein-kinase CK2 subunit interaction

Béatrice Laudet , Caroline Barette , Vincent Dulery , Olivier Renaudet , Pascal Dumy , et al.
Biochemical Journal, 2007, 408 (3), pp.363-373. ⟨10.1042/BJ20070825⟩
Journal articles hal-00478835v1
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Blockade of Platelet CysLT1R Receptor with Zafirlukast Counteracts Platelet Protumoral Action and Prevents Breast Cancer Metastasis to Bone and Lung

Lou Saier , Johnny Ribeiro , Thomas Daunizeau , Audrey Houssin , Gabriel Ichim , et al.
International Journal of Molecular Sciences, 2022, 23 (20), pp.12221. ⟨10.3390/ijms232012221⟩
Journal articles inserm-03847792v1
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Förster Resonance Energy Transfer Based Biosensor for Targeting the hNTH1–YB1 Interface as a Potential Anticancer Drug Target

Muge Senarisoy , Caroline Barette , Françoise Lacroix , Salvatore Debonis , Meike Stelter , et al.
ACS Chemical Biology, 2020, 15 (4), pp.990-1003. ⟨10.1021/acschembio.9b01023⟩
Journal articles cea-02517754v1

Pharmacological inhibition of LIM Kinase stabilizes microtubules and inhibits neoplastic growth

Renaud Prudent , Emilie Vassal-Stermann , Chi-Hung Nguyen , Catherine Pillet , Anne Martinez , et al.
Cancer Research, 2012, 72 (17), pp.4429-4439. ⟨10.1158/0008-5472.CAN-11-3342⟩
Journal articles hal-02348076v1